555 TERPENE CONJUGATION ACKNOWLEDGMENT This paper is a part of a PhD thesis by Seyedeh Maryam Mortazavi at the School of Pharmacy, Shahid Beheshti University of Medical Sciences (SBMU), Tehran, Iran and was financially supported by SBMU. REFERENCES (1) F. Gorouhi and H. I. Maibach, Role of topical peptides in preventing or treating aged skin, Int. J. Cosmet. Sci., 31, 327–345 (2009). (2) M. P. Lupo and A. L. Cole, Cosmeceutical peptides, Dermatol. Ther., 20, 34–349 (2007). (3) R. R. Jones, V. Castelletto, C. J. Connon, and I. W. Hamley, Collagen, Stimulating effect of peptide amphiphile C16–KTTKS on human fibroblasts, Mol. Pharm., 10, 1063–1069 (2013). (4) Y. L. Choi, E. J. Park, E. Kim, D. H. Na, and Y. H. Shin, Dermal stability and in vitro skin permeation of collagen pentapeptides (KTTKS and palmitoyl-KTTKS), Biomol. Ther., 22, 321–327 (2014). (5) C. Lu, B. M. Kim, D. Lee, M. h. Lee, J. h. Kim, H. b. Pyo, and K. Y. Chai, Synthesis of lipoic acid- peptide conjugates and their effect on collagen and melanogenesis, Eur. J. Med. Chem., 69, 449–454 (2013). (6) H. I. Choi, H. j. Kim, J. I. Park, E. H. Shin, D. W. Kim, and S. S. Kim, Design and efficient synthesis of novel ascorbyl conjugated peptide with high collagen biosynthesis stimulating effects, Bioorg. Med. Chem. Lett., 19, 2079–2082 (2009). (7) M. S. Kim, E. J. Park, and D. H. Na, Synthesis and characterization of monodisperse poly(ethylene glycol)-conjugated collagen pentapeptides with collagen biosynthesis-stimulating activity, Bioorg. Med. Chem. Lett., 25, 38–42 (2015). (8) D. A. Guglielmi, A. M. Martinelli, N. C. Rissi, E. M. Cilli, C. P. Soares, and L. A. Chiavacci, Synthesis of the peptide ac-wahx-kttks and evaluation of the ability to induce in vitro collagen synthesis, Protein. Pept. Lett., 23, 544–547 (2016). (9) J. P. Atkinson, H. I. Maibach, and N. Dragicevic, “Targets in dermal and transdermal delivery and classifi cation of penetration enhancement methods,” in: Percutaneous Penetration Enhancers Chemical Methods in Penetration Enhancement, N. Dragicevic-Curic, H. I. Maibach. Eds. (Springer-Verlag Berlin Heidelberg, Berlin 2015), pp. 102. (10) H. Moghimi, A. Williams, and B. Barry, A lamellar matrix model for stratum corneum intercellular lipids IV. Effects of terpene penetration enhancers on the permeation of 5-fluororacil and oestradiol through the matrix, Int. J. Pharm., 145, 49–59 (1996). (11) H. Moghimi, A. Williams, and B. Barry, A lamellar matrix model for stratum corneum intercellular lipids. V. Effects of terpene penetration enhancers on the structure and thermal behaviour of the matrix. Int. J. Pharm., 146, 41–54 (1997). (12) H. R. Moghimi, A. C. Williams, and B. W. Barry, A lamellar matrix model for stratum corneum intercellular lipids III. Effects of terpene penetration enhancers on the release of 5-fluorouracil and oestradiol from the matrix, Int. J. Pharm., 145, 37–47 (1996). (13) H. R. Moghimi, A. C. Williams, and B. W. Barry, Enhancement by terpenes of 5-fluorouracil permeation through the stratum corneum: model solvent approach. J. Pharm. Pharmacol., 50, 955–64 (1998). (14) S. M. Mortazavi, F. Kobarfard, H. I. Maibach, and H. R. Moghimi, Effect of palmitic acid conjugation on physicochemical properties of peptide KTTKS: A preformulation study. J. Cosmet. Sci., 70, 299–312 (2019). (15) F. Wohnsland and B. Faller, High-throughput permeability pH profile and high-throughput alkane/ water log P with artificial membranes, J. Med. Chem, 44, 923–930 (2001). (16) V. Kassis and J. Søndergaard, Heat separation of normal human skin for epidermal and dermal prostaglandin analysis, Arch. Dermatol. Res., 273, 301–306 (1982). (17) ACDLabs. ACD/ChemSketch.12.01 edn. Advanced Chemistry Development, Inc., Toronto, ON, Canada, www.acdlabs.com, 2009. (18) P. Palladino, V. Castelletto, A. Dehsorkhi, D. Stetsenko, and I. Hamley, Conformation and self-association of peptide amphiphiles based on the KTTKS collagen sequence, Langmuir, 28, 12209–12215 (2012). (19) H. R. Moghimi, A. C. Williams, and B. W. Barry, A lamellar matrix model for stratum corneum intercellular lipids. I. Characterisation and comparison with stratum corneum inter-cellular structure. Int. J. Pharm., 131, 103–115 (1996).
556 JOURNAL OF COSMETIC SCIENCE (20) A. Manafi, A. Hashemlou, P. Momeni, and H. R. Moghimi, Enhancing drugs absorption through third- degree burn wound eschar, Burns, 34, 698–702 (2008). (21) H. R. Moghimi, B. S. Makhmalzadeh, and A. Manafi, Enhancement effect of terpenes on silver sulphadiazine permeation through third-degree burn eschar, Burns, 35, 1165–1170 (2009). (22) H. R. Moghimi, F. H. Shirazi, M. Shafiee Ardestani, M. A. Oghabian, M. Saffari, and J. Sojoudi, In vitro and in vivo enhancement of antitumoral activity of liposomal antisense oligonucleotides by cineole as a chemical penetration enhancer, J. Nanomater, 2015, 10 (2015).
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